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Cayman Chemical SB-243213hydrochlorIde 5mg
Supplier: Cayman Chemical 362175 MG
A 5-HT2C receptor inverse agonist; selective for 5-HT2C over the 5-HT2A and 5-HT2B receptors (Kis = 0.001, 0.158, and 0.1 µM, respectively) and CYP1A2, CYP2C9, CYP2C19, CYP2D6, and CYP3A4 (IC50s = >100, 23, >100, >100, and >100 µM, respectively); reduces the basal activity of 5-HT2C in HEK293 cells expressing the human receptor (pKB = 9.5); reverses mCPP-induced hypolocomotion in rats (ID50 = 0.7 mg/kg); has anxiolytic-like activity in the social interaction test in rats at 0.2-5 mg/kg
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