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Medchemexpress LLC SB 271046 Hydrochloride | 209481-24-3 | 99.9% | C20H23Cl2N3O3S2 | 50 MG
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Supplier:  Medchemexpress LLC HY14336A50MG

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SB 271046 Hydrochloride is a potent, selective, orally active, and BBB-permeable 5-HT6 receptor antagonist. It exhibits high selectivity for the 5-HT6 receptor compared to 55 other receptors, binding sites, and ion channels, and also demonstrates anticonvulsant activity.

  • Potent, selective, orally active, and BBB-permeable 5-HT6 receptor antagonist
  • Over 200-fold selectivity for the 5-HT6 receptor
  • Shows anticonvulsant activity (EC50=0.16 μM)
  • Antagonizes 5-HT-induced stimulation of adenylyl cyclase activity (pA2=8.71)
  • Increases seizure threshold in rat maximal electroshock seizure threshold (MEST) test in vivo

Catalog No. 50-003-55014


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