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Medchemexpress LLC Talabostat (mesylate) | 150080-09-4 | 98.4% | 310.18 | 5 MG
Supplier: Medchemexpress LLC 5MGHY13233A
Talabostat mesylate is an orally active and nonselective dipeptidyl peptidase IV (DPP-IV) inhibitor and an inhibitor of fibroblast activation protein (FAP). It also inhibits other DASH family enzymes and exhibits antineoplastic and hematopoiesis-stimulating activities.
- Orally active and nonselective DPP-IV inhibitor (IC50 < 4 nM; Ki = 0.18 nM)
- Inhibitor of fibroblast activation protein (FAP) (IC50 = 560 nM)
- Inhibits DPP8/9 (IC50 = 4/11 nM; Ki = 1.5/0.76 nM), quiescent cell proline dipeptidase (QPP) (IC50 = 310 nM), and DPP2
- Exhibits antineoplastic and hematopoiesis-stimulating activities
- Stimulates immune responses against tumors involving both innate and adaptive immune systems
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