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Medchemexpress LLC TC-2559 difumarate | 2454492-41-0 | 98.4% | 438.43 | 1 MG
Supplier: Medchemexpress LLC HY1362071MG
TC-2559 difumarate is a central nervous system (CNS)-selective, orally active partial agonist of the α4β2 subtype of nicotinic acetylcholine receptors (nAChR).
- Selectivity for α4β2 receptors over α2β4, α4β4, and α3β4 receptors, with EC50 values ranging from 10-30 μM.
- Demonstrates an antinociceptive effect, reducing formalin-induced nociceptive responses in mice and inhibiting chronic constriction injury-induced neuropathic pain in rats.
- Solubility of 43.84 mg/mL (99.99 mM) in H2O, requiring ultrasonic and warming for preparation.
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