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Medchemexpress LLC Thiq | 312637-48-2 | MFCD09970598 | 98.5% | 589.17 | C33H41ClN6O2 | 10 MG
Supplier: Medchemexpress LLC HY1062410MG
THIQ is a selective melanocortin-4 receptor (MC4R) agonist used in research to probe MC4R signaling and receptor trafficking. It functions as a pharmacoperone that can rescue cell-surface expression and signaling of certain intracellularly retained MC4R mutants and has been employed in rodent studies of erectile activity.
- Selective MC4R agonist with high affinity and potency (hMC4R IC50=1.2 nM; EC50=2.1 nM; rMC4R IC50=0.6 nM; EC50=2.9 nM).
- Acts as a pharmacoperone to restore receptor cell-surface expression.
- High reported purity and supplied as a solid, white to off-white material.
- Stable under recommended storage (powder: -20°C for 3 years; 4°C for 2 years).
- Suitable for in vitro and in vivo studies of melanocortin receptor biology.
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