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Medchemexpress LLC Zen-2759 | 1616400-50-0 | 99.5% | 280.32 g·mol⁻¹ | C17H16N2O2 | 5 MG

Supplier: Medchemexpress LLC HY1292015MG
ZEN-2759 is a research-grade small-molecule BET (bromodomain and extra-terminal) inhibitor that selectively targets BRD4 bromodomains. Reported biochemical potency includes IC50 values of 0.23 μM (BRD4 BD1), 0.08 μM (BRD4 BD2), and 0.28 μM (BRD4 BD1BD2). The compound is supplied as a purified solid for in vitro laboratory research and is not for human or diagnostic use.
- Potent inhibition of BRD4 bromodomains at submicromolar concentrations.
- Well-characterized activity with reported IC50 values for BD1, BD2, and BD1BD2.
- Supplied as a high-purity research compound suitable for biochemical assays.
- Includes analytical data supporting identity and purity.
- Useful tool for epigenetic and transcriptional regulation studies in vitro.
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