Oxazinanes
Selleck Chemical LLC Moxisylyte hydrochloride
Moxisylyte hydrochloride (thymoxamine) is an alpha-adrenergic blocking agent used for the treatment of Raynaud s disease
Selleck Chemical LLC Triflupromazine hydrochloride
Triflupromazine hydrochloride (Fluopromazine) is an antipsychotic medication of the phenothiazine class
(N)C1 | 100mg | 808545143](https://assets.fishersci.com/TFS-Assets/CCG/product-images/502694492.jpg-250.jpg)
eMolecules 1817789-07-3 | tert-butyl (3R)-3-amino-3-methylpyrrolidine-1-carboxylate | Synthonix | MFCD30471114 | 200.282 | C10H20N2O2 | 97.000 | CC(C)(C)OC(=O)N1CC[C@@](C)(N)C1 | 100mg | 808545143
tert-butyl (3R)-3-amino-3-methylpyrrolidine-1-carboxylate | Synthonix | 1817789-07-3 | MFCD30471114 | 200.282 | C10H20N2O2 | 97.000 | CC(C)(C)OC(=O)N1CC[C@@](C)(N)C1 | 100mg | 808545143
Apexbio Technology LLC Sarpogrelate hydrochloride 135159-51-2 10mM (in 1mL DMSO)
Sarpogrelate hydrochloride (CAS 135159-51-2) is a selective antagonist of the 5-HT2A receptor exhibiting a binding affinity (Ki) of 8 39 nM comparable to ritanserin By inhibiting 5-HT2A receptor-mediated pathways sarpogrelate suppresses platelet aggregation thrombus formation and vascular smooth muscle cell proliferation In vitro its primary metabolite (M-1) blocks 5-HT-induced responses at the 5-HT2A receptor with minimal stereoselective difference Clinically oral administration of sarpogrelate in patients with peripheral arterial disease significantly enhances forearm and leg blood flow responses to reactive hyperemia indicating improved vascular function Sarpogrelate is employed in research on platelet function thrombosis and vascular disorders
Cayman Chemical 3-OxocholIc AcId 250mg
A secondary bile acid; a metabolite of cholic acid in C. perfringens; serum levels increase following ileal transposition surgery in rats
Selleck Chemical LLC GPNA hydrochloride
GPNA hydrochloride (L- -glutamyl-p-nitroanilide hydrochloride) is a substrate of -glutamyltransferase (GGT) and an inhibitor of the glutamine transporter ASCT2 with an IC50 of 250 M in A549 cells It also inhibits Na -dependent carriers SNAT1 -2 -4 -5 and Na -independent leucine transporters LAT1/2 It can be widely used in research on pancreatic cancer breast cancer glioblastoma multiforme acute myelogenous leukemia and non-small-cell lung cancer
Medchemexpress LLC m-PEG6-Br | 125562-29-0 | 99.8% | C13H27BrO6 | 250 MG
m-PEG6-Br is a PEG-based PROTAC linker used in the synthesis of PROTACs. PROTACs leverage the intracellular ubiquitin-proteasome system to selectively degrade target proteins, by connecting an E3 ubiquitin ligase ligand to a target protein ligand via a linker.
- Used in the synthesis of PROTACs
- Exploits the intracellular ubiquitin-proteasome system
- Selectively degrades target proteins
- Pure form storage: -20°C for 3 years, 4°C for 2 years
- In solvent storage: -80°C for 6 months, -20°C for 1 month
TARGETMOL CHEMICALS INC SKF-34288 HYDROCHLORIDE 5MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg and bulk. Please contact Fisher for quotes. SKF-34288 hydrochloride (3-Mercaptopicolinic acid hydrochloride) is an inhibitor of phosphoenolpyruvate carboxykinase (PEPCK)and inhibits Asn metabolism and results in an increase in amino acids and amides. purity: 95%
TARGETMOL CHEMICALS INC SRT1720 HYDROCHLORIDE 5MG
Also available in 1 mg 2 mg 10 mg 25 mg 50 mg 100 mg 200 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. SRT1720 hydrochloride (SRT1720 HCl) is a selective activator of SIRT1 (EC1.5 0.16 uM) and shows less potent activities on SIRT2/SIRT3 (EC1.5s 37 uM/300 uM). purity: 99%
TARGETMOL CHEMICALS INC PONATINIB HYDROCHLORIDE 10MG
Also available in 25 mg 50 mg 100 mg 200 mg 500 mg and bulk. Please contact Fisher for quotes. Ponatinib Hydrochloride (AP-24534 Hydrochloride) is a hydrochloride of ponatinib. Ponatinib is an orally active multi-targeted kinase inhibitor with IC50s of 0.37 nM 1.1 nM 1.5 nM 2.2 nM and 5.4 nM for Abl PDGFR(alpha) VEGFR2 FGFR1 and Src respectively. purity: 100%
TARGETMOL CHEMICALS INC SALUBRINAL 25MG
Also available in 2 mg 5 mg 10 mg 50 mg 100 mg 500 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. Salubrinal a phosphatases (PP1) inhibitor(IC50=1.7 uM) exhibits function on the eukaryotic translation initiation factor 2 subunit (eIF2(alpha)). purity: 99%