CAS RN 1333377-65-3
CAS RN 1333377-65-3
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MilliporeSigma™ Calbiochem™ Haspin Kinase Inhibitor, CHR-6494
A cell-permeable indazolylimidazopyridazinamine compound that acts as a potent and reversible inhibitor of histone kinase haspin activity (IC50 = 2nM) with moderate selectivity over TrkA, GSK-3β, PIM1, Cdk1/B and Cdk2/A (% inhibition at 100nM = 58, 48, 36, 34 and 33, respectively) among a panel of 27-kina