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Medchemexpress LLC 1H-Benzimidazole, 2-[[2-(4-chlorophenoxy)ethyl]thio]- | 312749-73-8 | 99.9% | C15H13ClN2OS | 1 ML
SDP

Catalog No. 5000353433
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CLP-3094 is a potent BF3 (binding function 3)-directed inhibitor of the androgen receptor (AR), inhibiting its transcriptional activity with an IC50 of 4 μM. It also acts as a selective and potent GPR142 antagonist.

  • Potent BF3-directed inhibitor of androgen receptor (AR)
  • Inhibits AR transcriptional activity (IC50=4 μM)
  • Selective, potent GPR142 antagonist
  • Inhibits increase of intracellular Ca2+ concentration induced by L-tryptophan in CHO-K1 cells expressing GPR142
  • Inhibits accumulation of inositol phosphates in HEK293 cells expressing GPR142
  • Inhibits insulin secretion from islets induced by L-tryptophan and GPR142 agonists
  • For research use only

Catalog No. 50-003-53433 Supplier Medchemexpress LLC Supplier No. HY14148710MM/1ML
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CLP-3094 is a potent BF3 (binding function 3)-directed inhibitor of the androgen receptor (AR), inhibiting its transcriptional activity with an IC50 of 4 μM. It also acts as a selective and potent GPR142 antagonist.

  • Potent BF3-directed inhibitor of androgen receptor (AR)
  • Inhibits AR transcriptional activity (IC50=4 μM)
  • Selective, potent GPR142 antagonist
  • Inhibits increase of intracellular Ca2+ concentration induced by L-tryptophan in CHO-K1 cells expressing GPR142
  • Inhibits accumulation of inositol phosphates in HEK293 cells expressing GPR142
  • Inhibits insulin secretion from islets induced by L-tryptophan and GPR142 agonists
  • For research use only

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