Promotional price valid on web orders only. Your contract pricing may differ. Interested in signing up for a dedicated account number?
Learn More
  1. Home
  2. Products
  3. 5000339771

Medchemexpress LLC 2H-1,2,4-Benzothiadiazine, 4-cyclopropyl-7-fluoro-3,4-dihydro-, 1,1-dioxide | 1204572-55-3 | 99.7% | 100 MG
SDP

Supplier:  Medchemexpress LLC HY129086100MG

Encompass_Preferred

BPAM344 is a positive allosteric modulator (PAM) of kainate receptor (KAR) subunits GluK1b, GluK2a, and GluK3a, primarily used for research. It potentiates glutamate-evoked currents of GluK2a and significantly decreases desensitization kinetics. It also modulates AMPA receptor activity in primary neuron cell cultures.

  • Positive allosteric modulator of KAR subunits GluK1b, GluK2a, GluK3a
  • Potentiates glutamate-evoked currents of GluK2a (EC50 of 79 μM)
  • Decreases desensitization kinetics (5.5 to 775 ms)
  • Potentiates peak current amplitude of KAR and AMPA receptor subunits
  • Modulates AMPA receptor in rat embryonic cortex primary neuronal culture (EC50 of 0.9 μM)
  • Molecular weight: 242.27
  • Chemical formula: C10H11FN2O2S
  • Appearance: White to off-white solid

Catalog No. 50-003-39771


May include imposed supplier surcharges.
Add to Cart

Product Title
Select an issue

By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.