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Medchemexpress LLC 3-cyclopropyl-1-[[4-[6-[(1,1-dioxo-1,4-thiazinan-4-yl)methyl]-5-fluoropyridin-2-yl]phenyl]methyl]imi | 2250025-91-1 | Not found | 99.4% | 508.99 | C23H25FN4O4S·HCl | 25MG

Supplier: Medchemexpress LLC HY124283A25MG
LEI-101 hydrochloride is a potent, selective, orally bioavailable cannabinoid CB2 receptor agonist supplied for research use. It demonstrates strong functional activity at human CB2 receptors with substantially lower affinity for CB1 and minimal hERG binding, suitable for in vitro and in vivo pharmacology studies.
- Purity 99.4%.
- Reported activity pEC50 = 8 for human CB2.
- Approximately 100-fold selectivity for CB2 over CB1.
- Low hERG interaction (pKi < 4).
- Soluble in DMSO; available as dry powder and 10 mM solution in DMSO.
- Intended for research use only; not for human or clinical use.
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