Promotional price valid on web orders only. Your contract pricing may differ. Interested in signing up for a dedicated account number?
Learn More

Medchemexpress LLC 3-cyclopropyl-1-[[4-[6-[(1,1-dioxo-1,4-thiazinan-4-yl)methyl]-5-fluoropyridin-2-yl]phenyl]methyl]imi | 2250025-91-1 | Not found | 99.4% | 508.99 | C23H25FN4O4S·HCl | 25MG
SDP

Supplier:  Medchemexpress LLC HY124283A25MG

Encompass_Preferred

LEI-101 hydrochloride is a potent, selective, orally bioavailable cannabinoid CB2 receptor agonist supplied for research use. It demonstrates strong functional activity at human CB2 receptors with substantially lower affinity for CB1 and minimal hERG binding, suitable for in vitro and in vivo pharmacology studies.

  • Purity 99.4%.
  • Reported activity pEC50 = 8 for human CB2.
  • Approximately 100-fold selectivity for CB2 over CB1.
  • Low hERG interaction (pKi < 4).
  • Soluble in DMSO; available as dry powder and 10 mM solution in DMSO.
  • Intended for research use only; not for human or clinical use.

Catalog No. 50-002-36923


May include imposed supplier surcharges.
Only null left
Add to Cart

Product Title
Select an issue

By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.