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Medchemexpress LLC 4-(4-((dimethylamino)methyl)-2,5-dimethoxyphenyl)-2-methyl-2,7-naphthyridin-1(2H)-one | 1883429-22-8 | >98.0% | 353.17 Da | C20H23N3O3 | 100 MG
SDP

Supplier:  Medchemexpress LLC HY100352100MG

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BI-9564 is a potent, selective, and cell-permeable small-molecule inhibitor of the BRD9 bromodomain, with weaker activity against BRD7. Developed through structure-guided design, it binds BRD9 in the low-nanomolar range and has been used as a chemical probe in cellular assays and in vivo studies, including reported oral efficacy in preclinical AML models.

  • High affinity for BRD9 with weaker activity against BRD7.
  • Demonstrated cellular potency (AlphaScreen IC50 ≈ 75 nM).
  • Cell-permeable and suitable for cellular and in vivo studies.
  • Validated structural data available (PDB: 5F1H).
  • Useful as a research chemical probe to study chromatin remodeling biology.
  • Available from multiple research suppliers in small-mass packaging.

Catalog No. 50-002-12676


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