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Medchemexpress LLC 4-[6-[[4-(cyclopropylmethyl)piperazin-1-yl]methyl]-2-(5-fluoro-1H-indol-4-yl)thieno[3,2-d]pyrimidin- | 955977-50-1 | 99.0% | 10 MG

Supplier: Medchemexpress LLC HY1223510MG
PI-3065 is a selective small-molecule inhibitor of the PI3K p110δ isoform with potent biochemical inhibition and characterized isoform selectivity. It is supplied as a powder for research use.
- Potent inhibition of PI3K p110δ (IC50 5 nM; Ki 1.5 nM).
- Markedly reduced activity against p110α, p110β, and p110γ (IC50s 910 nM, 600 nM, >10,000 nM).
- Provided as a powder in 10 MG quantities.
- Powder storage: stable at -20°C (3 years) and 4°C (2 years) when stored as recommended.
- Demonstrated activity in cellular and in vivo models consistent with p110δ targeting.
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