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Medchemexpress LLC 4H-1-Benzopyran-4-one, 6-methoxy-5-nitro-2-(trifluoromethyl)- | 342795-08-8 | 99.85% | 289.16 | 50 MG
SDP

Supplier:  Medchemexpress LLC HY11155010MG

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Bragsin2 is a potent, selective, and noncompetitive nucleotide exchange factor BRAG2 inhibitor with an IC50 of 3 μM. It binds at the interface between the PH domain of BRAG2 and the lipid bilayer, preventing activation of lipidated Arf GTPase. This compound affects breast cancer stem cells.

  • Potent, selective, and noncompetitive nucleotide exchange factor BRAG2 inhibitor with an IC50 of 3 μM.
  • Binds at the interface between the PH domain of BRAG2 and the lipid bilayer.
  • Leads to BRAG2 being unable to activate lipidated Arf GTPase.
  • Affects breast cancer stem cells.
  • Inhibits Arf GTPase activation in HeLa cells at 50 μM.
  • Inhibits the growth of SUM149 and S68 cells at 50 μM.

Catalog No. 50-003-46573


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