Medchemexpress LLC 6-[[4-(cyclopropylmethyl)-1-piperazinyl]methyl]-2-(5-fluoro-indol-4-yl)-4-(4-morpholinyl)-thieno-pyrimidine | 955977-50-1 | 99.0% | 50 MG

Supplier:  Medchemexpress LLC HY1223550MG

PI-3065 is a selective small-molecule inhibitor of PI3K p110δ used for research applications. It potently inhibits p110δ (IC50 5 nM; Ki 1.5 nM) and shows substantially lower activity against other PI3K isoforms, and is supplied as a solid for in vitro and in vivo studies.

• Potent p110δ inhibition (IC50 5 nM; Ki 1.5 nM).
• Reduced activity against p110α (IC50 910 nM), p110β (IC50 600 nM), p110γ (>10,000 nM).
• Purity approximately 98.97%.
• Chemical formula C27H31FN6OS; molecular weight 506.64 g/mol.
• Appearance: white to off-white solid.
• Soluble in DMSO (25 mg/mL) and formulatable for in vivo dosing.
• Storage: powder -20°C (up to 3 years) or 4°C (up to 2 years).
• Available in small-mass pack sizes (for example 50 mg).

Catalog No. 50-002-30705