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Medchemexpress LLC 6,7-dimethoxy-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine | 319492-82-5 | 98.8% | 370.405 | C20H22N2O5 | 50MG

Supplier: Medchemexpress LLC HY12479350MG
GAK inhibitor 49 is a potent, ATP-competitive, and highly selective inhibitor of cyclin G-associated kinase (GAK) used as a research tool to probe GAK-related signaling. It exhibits sub-nanomolar binding affinity and low-nanomolar cellular potency, and is provided as a high-purity solid for in vitro studies.
- Potent ATP-competitive inhibition of GAK (Ki = 0.54 nM).
- High cellular potency suitable for cell-based assays (cell IC50 = 56 nM).
- High purity for biochemical testing (>98%).
- Well characterized molecular properties (MW 370.40 g/mol; C20H22N2O5).
- Available in small research quantities for assay development and screening.
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