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TARGETMOL CHEMICALS INC A-366 25MG
SDP

Supplier:  TARGETMOL CHEMICALS INC T362425MG

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Also available in 1 mg 2 mg 5 mg 10 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. A-366 is a highly selective peptide-competitive histone methyltransferase G9a inhibitor with IC50s of 3.3 and 38 nM for G9a and GLP respectively.It is more than 1000-fold selective for G9a and GLP over the other 21 methyltransferases. It is an inhibitor of the Spindlin1-H3K4me3 interaction with an IC50 of 182.6 nM.It exhibits high affinity for human H3R with a Ki value of 17 nM and shows subtype selectivity between subgroups of the histaminergic and dopaminergic receptor families. purity: 99%

Catalog No. 50-258-0194


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