Promotional price valid on web orders only. Your contract pricing may differ. Interested in signing up for a dedicated account number?
Learn More
Learn More
Medchemexpress LLC ADL-5859 (hydrochloride) | 850173-95-4 | 99.0% | 25 MG
Supplier: Medchemexpress LLC 25MGHY13044
ADL-5859 hydrochloride is a selective and orally active δ opioid receptor (DOR) agonist with a Ki of 0.84 nM and an EC50 value of 20 nM. It also exhibits inhibitory activity to the hERG channel with an IC50 value of 78 μM. This compound is suitable for pain research.
- Selective and orally active δ opioid receptor (DOR) agonist
- Ki of 0.84 nM and EC50 of 20 nM for δ opioid receptor
- Inhibits hERG channel with IC50 of 78 μM
- Inhibits cytochrome P450 2D6 (CYP2D6) with IC50 of 43 μM
- Suitable for pain research
- Reverses hyperalgesia in the inflamed paw of rats
- Shows antidepressant-like activity in rats
- Appears as a white to off-white solid
- Molecular weight: 428.95
- Chemical formula: C24H29ClN2O3
Product Title
By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.
Spot an opportunity for improvement?