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Medchemexpress LLC AKR1C1-IN-1 | 4906-68-7 | 99.4% | 293.11 | 10 MG
Supplier: Medchemexpress LLC HY11400910MG
AKR1C1-IN-1 is a potent and selective inhibitor of human 20α-hydroxysteroid dehydrogenase (AKR1C1), demonstrating a a Ki value of 4 nM for AKR1C1. It is intended for research use only.
- Ki value for AKR1C1: 4 nM
- Inhibition of AKR1C2: 87 nM
- Inhibition of AKR1C3: 4.2 μM
- Inhibition of AKR1C4: 18.2 μM
- Potently inhibits the metabolism of progesterone in AKR1C1-overexpressed BAECs, with an IC50 of 460 nM.
- Target: Aldose Reductase
- Pathway: Metabolic Enzyme/Protease
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