Promotional price valid on web orders only. Your contract pricing may differ. Interested in signing up for a dedicated account number?
Learn More

AM 281, Tocris Bioscience™

Click to view available options
Quantity:
10mg
50mg
202463-68-1
C21H19Cl2IN4O2
557.213
AJFFBPZYXRNAIC-UHFFFAOYSA-N
unii-sbp4a4dyh2,sbp4a4dyh2,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-4-morpholinyl-1h-pyrazole-3-carboxamide,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-morpholin-4-ylpyrazole-3-carboxamide,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-morpholino-1h-pyrazole-3-carboxamide,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-morpholin-4-yl pyrazole-3-carboxamide,tocris-1115,d0ud9h,gtpl741,1h-pyrazole-3-carboxamide, 1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-4-morpholinyl
4302962
1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-morpholin-4-ylpyrazole-3-carboxamide
CC1=C(N(N=C1C(=O)NN2CCOCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)I
202463-68-1
C21H19Cl2IN4O2
557.213
AJFFBPZYXRNAIC-UHFFFAOYSA-N
unii-sbp4a4dyh2,sbp4a4dyh2,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-4-morpholinyl-1h-pyrazole-3-carboxamide,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-morpholin-4-ylpyrazole-3-carboxamide,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-morpholino-1h-pyrazole-3-carboxamide,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-morpholin-4-yl pyrazole-3-carboxamide,tocris-1115,d0ud9h,gtpl741,1h-pyrazole-3-carboxamide, 1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-4-morpholinyl
4302962
1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-morpholin-4-ylpyrazole-3-carboxamide
CC1=C(N(N=C1C(=O)NN2CCOCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)I

Potent, selective CB1 antagonist/inverse agonist

Potent, selective CB 1 cannabinoid receptor antagonist/inverse agonist (K i values are 12 and 4200 nM for CB 1 and CB 2 receptors respectively). Increases locomotor activity following systemic administration in vivo. Analog of SR141716A (K i = 14 nM).
Quantity 50mg
Formula Weight 557.22
Percent Purity >99%
Chemical Name or Material AM 281

Recommended Storage : Desiccate at +4°C