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Cayman Chemical RF9, Purity: ≥98%, CAS: 876310-60-0, 10 mg
SDP

Catalog No. 502991694
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An NPFF receptor antagonist; binds to human NPFF1 and NPFF2 receptors (Kis = 58 and 75 nM, respectively); selective for NPFF1 and NPFF2 receptors over NPY receptor Y1, GPR10, GPR54, GPR103, ORL-1, and μ-, δ-, and κ-opioid receptors at 10 μM; inhibits NPFF-induced [35S]GTPγS binding to the NPFF2 receptor at 7.5 μM; reverses NPVF-induced inhibition of forskolin-stimulated cAMP accumulation in CHO cells expressing the human NPFF1 receptor (EC50 = 4.7 μM); inhibits NPFF-induced increases in mean arterial pressure and heart rate in rats at 10 μg, i.c.v.; prevents heroin-induced delayed hyperalgesia and associated tolerance in rats at 0.1 mg/kg, s.c.

Catalog No. 50-299-1694 Supplier Cayman Chemical Supplier No. 3141210 MG
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An NPFF receptor antagonist; binds to human NPFF1 and NPFF2 receptors (Kis = 58 and 75 nM, respectively); selective for NPFF1 and NPFF2 receptors over NPY receptor Y1, GPR10, GPR54, GPR103, ORL-1, and μ-, δ-, and κ-opioid receptors at 10 μM; inhibits NPFF-induced [35S]GTPγS binding to the NPFF2 receptor at 7.5 μM; reverses NPVF-induced inhibition of forskolin-stimulated cAMP accumulation in CHO cells expressing the human NPFF1 receptor (EC50 = 4.7 μM); inhibits NPFF-induced increases in mean arterial pressure and heart rate in rats at 10 μg, i.c.v.; prevents heroin-induced delayed hyperalgesia and associated tolerance in rats at 0.1 mg/kg, s.c.

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