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Medchemexpress LLC Azasetron hydrochloride | 123040-16-4 | 99.8% | C17H21Cl2N3O3 | 100 MG
SDP

Supplier:  Medchemexpress LLC HYB0068100MG

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Azasetron hydrochloride is a benzamide derivative that functions as a potent and selective antagonist of the 5-HT3 receptor, demonstrating an IC50 of 0.33 nM against this target. It has been investigated for its potential in studies related to chemotherapy-induced nausea and vomiting (CINV) and has shown the ability to penetrate the skin and enter systemic circulation in in vivo models.

  • Mechanism of action: Potent and selective 5-HT3 receptor antagonist.
  • Target affinity: IC50 of 0.33 nM for 5-HT3 receptor.
  • Chemical classification: Benzamide derivative.
  • Molecular formula: C17H21Cl2N3O3.
  • Molecular weight: 386.27.
  • Purity: 99.76%.
  • Physical characteristics: White to off-white solid.
  • Solubility: Soluble in water (20 mg/mL) and DMSO (2.22 mg/mL).
  • Research application: Used in CINV studies.
  • Pharmacokinetic property: Penetrates skin and enters systemic circulation in animal models.

Catalog No. 50-004-32157


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