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Medchemexpress LLC Benzo[lmn]phenanthroline-1,3,6,8(2H,7H)-tetrone, 2,7-bis(4-hydroxybutyl)- | 298217-59-1 | C22H22N2O6 | 5 MG
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Catalog No. 5000373745
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MMV009085 is a potent Plasmodium falciparum hexose transporter (PfHT1)-specific inhibitor and a potential anti-malarial agent. It also acts as a human glucose transporter inhibitor, demonstrating high potency in inhibiting both glucose uptake (IC50: 2.6 μM) and the growth of parasites (EC50: 1.23 ± 0.04 μM against 3D7).

  • Potent PfHT1-specific inhibitor
  • Potential anti-malarial agent
  • Human glucose transporter inhibitor
  • High potency in inhibiting glucose uptake (IC50: 2.6 μM)
  • Inhibits growth of various parasite strains (EC50: 1.23 ± 0.04 μM; 0.720 ± 0.05 μM)
  • Inhibits transport activity of PfHT-1 (IC50: 212 ± 39 μM)
  • Shows cytotoxicity against HEK293T cells (CC50: 2.46 ± 0.03 μM) and HepG2 cells (CC50: 1.92 ± 0.85 μM)
  • Acts through PfHT blockage to inhibit parasite growth (EC50 = 0.795 μM)

Catalog No. 50-003-73745 Supplier Medchemexpress LLC Supplier No. HY1536125MG
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MMV009085 is a potent Plasmodium falciparum hexose transporter (PfHT1)-specific inhibitor and a potential anti-malarial agent. It also acts as a human glucose transporter inhibitor, demonstrating high potency in inhibiting both glucose uptake (IC50: 2.6 μM) and the growth of parasites (EC50: 1.23 ± 0.04 μM against 3D7).

  • Potent PfHT1-specific inhibitor
  • Potential anti-malarial agent
  • Human glucose transporter inhibitor
  • High potency in inhibiting glucose uptake (IC50: 2.6 μM)
  • Inhibits growth of various parasite strains (EC50: 1.23 ± 0.04 μM; 0.720 ± 0.05 μM)
  • Inhibits transport activity of PfHT-1 (IC50: 212 ± 39 μM)
  • Shows cytotoxicity against HEK293T cells (CC50: 2.46 ± 0.03 μM) and HepG2 cells (CC50: 1.92 ± 0.85 μM)
  • Acts through PfHT blockage to inhibit parasite growth (EC50 = 0.795 μM)

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