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Medchemexpress LLC BI-3663 | 2341740-84-7 | 99.8% | 917.84 | 100 MG
Supplier: Medchemexpress LLC HY11154650MG
BI-3663 is a highly selective PTK2/FAK PROTAC (DC50=30 nM) that utilizes Cereblon ligands to hijack E3 ligases for PTK2 degradation. It inhibits PTK2 with an IC50 of 18 nM. BI-3663 is composed of BI-4464 (HY-124625) linked to Pomalidomide (HY-10984) with a linker, and demonstrates anti-cancer activity.
- Highly selective PTK2/FAK PROTAC
- Inhibits PTK2 with an IC50 of 18 nM
- Utilizes Cereblon ligands for PTK2 degradation
- Composed of BI-4464 linked to Pomalidomide with a linker
- Exhibits anti-cancer activity
- Potently degrades PTK2 in Hep3B2.1-7 cells and A549 cells
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