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Medchemexpress LLC BI-4020 | 2664214-60-0 | 99.3% | 1 ML
Supplier: Medchemexpress LLC HY12955010MM/1ML
BI-4020 is a fourth-generation, orally active, and non-covalent EGFR tyrosine kinase inhibitor. It shows activity against various EGFR variants, including the triple mutant EGFR del19 T790M C797S, the double mutant EGFR del19 T790M, and primary mutant EGFR del19. It also exhibits activity against EGFR wt.
- Inhibits EGFR del19 T790M C797S variant with an IC50 of 0.2 nM
- Inhibits EGFR del19 T790M and EGFR del19 with an IC50 of 1 nM
- Exhibits high kinome selectivity
- Possesses good DMPK properties
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