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Medchemexpress LLC BIX-01294 | 935693-62-2 | 98.4% | 490.64 | 250 MG
Supplier: Medchemexpress LLC 250MGHY10587
BIX-01294 is a reversible and highly selective G9a and GLP Histone Methyltransferase inhibitor, with IC50s of 1.7 μM and 0.9 μM, respectively. It inhibits G9a/GLP by competing for binding with the amino acids N-terminal of the substrate lysine residue. This (1H-1,4-diazepin-1-yl)-quinazolin-4-yl amine derivative induces necroptosis and autophagy and has antitumor activity in recurrent tumor cells.
- Reversible and highly selective G9a and GLP Histone Methyltransferase inhibitor
- Induces necroptosis and autophagy
- Exhibits antitumor activity in recurrent tumor cells
- Inhibits G9a/GLP by competing for binding with amino acids N-terminal of substrate lysine residue
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