Cayman Chemical BNTXmaleate 10mg

Supplier:  Cayman Chemical 3982910 MG

A δ1-opioid receptor antagonist (Ki = 0.1 nM); selective for the δ1-opioid receptor over the δ2-, μ-, and κ-opioid receptors (Kis = 10.8, 13.3, and 58.6 nM, respectively); decreases proliferation of primary mouse splenic B cells and the production of IL-2 and IL-4 by primary mouse splenic T lymphocytes at 1 and 10 µM; has antinociceptive activity in the tail-flick test in mice (ED50 = 46.4 pmol/animal) and decreases the antinociceptive activity of DPDPE at 6.3 pmol/animal; decreases the number of capsaicin-induced coughs in mice at 0.3-3 mg/kg; reduces the number of parasitized red blood cells in a mouse model of chloroquine-resistant P. chabaudi infection at 10 mg/kg

Catalog No. 50-297-8654