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Medchemexpress LLC Bragsin1 | 369631-68-5 | 99.9% | 273.16 | 10 MG
SDP

Supplier:  Medchemexpress LLC HY11154950MG

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Bragsin1 is a potent, selective, and noncompetitive inhibitor of the ArfGEF BRAG2, which inhibits Arf GTPase activation with an IC50 of 3 μM. It functions as a noncompetitive interfacial inhibitor by binding to the PH domain of BRAG2 and does not affect the Sec7 domain of human ArfGEFs. Bragsin1 also exhibits anti-cancer activity.

  • Potent, selective, and noncompetitive inhibitor of ArfGEF BRAG2.
  • Inhibits Arf GTPase activation with an IC50 of 3 μM.
  • Binds to the PH domain of BRAG2.
  • No effect on the Sec7 domain of human ArfGEFs.
  • Exhibits anti-cancer activity.

Catalog No. 50-003-46977


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