Promotional price valid on web orders only. Your contract pricing may differ. Interested in signing up for a dedicated account number?
Learn More
  1. Home
  2. Products
  3. 5000346977

Medchemexpress LLC Bragsin1 | 369631-68-5 | 99.9% | 273.16 | 10 MG
SDP

Catalog No. 5000346977
Encompass_Preferred

Bragsin1 is a potent, selective, and noncompetitive inhibitor of the ArfGEF BRAG2, which inhibits Arf GTPase activation with an IC50 of 3 μM. It functions as a noncompetitive interfacial inhibitor by binding to the PH domain of BRAG2 and does not affect the Sec7 domain of human ArfGEFs. Bragsin1 also exhibits anti-cancer activity.

  • Potent, selective, and noncompetitive inhibitor of ArfGEF BRAG2.
  • Inhibits Arf GTPase activation with an IC50 of 3 μM.
  • Binds to the PH domain of BRAG2.
  • No effect on the Sec7 domain of human ArfGEFs.
  • Exhibits anti-cancer activity.

Catalog No. 50-003-46977 Supplier Medchemexpress LLC Supplier No. HY11154950MG
May include imposed supplier surcharges.
Add to Cart
Add to Cart

Bragsin1 is a potent, selective, and noncompetitive inhibitor of the ArfGEF BRAG2, which inhibits Arf GTPase activation with an IC50 of 3 μM. It functions as a noncompetitive interfacial inhibitor by binding to the PH domain of BRAG2 and does not affect the Sec7 domain of human ArfGEFs. Bragsin1 also exhibits anti-cancer activity.

  • Potent, selective, and noncompetitive inhibitor of ArfGEF BRAG2.
  • Inhibits Arf GTPase activation with an IC50 of 3 μM.
  • Binds to the PH domain of BRAG2.
  • No effect on the Sec7 domain of human ArfGEFs.
  • Exhibits anti-cancer activity.

Product Title
Select an issue

By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.