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Medchemexpress LLC Bromocriptine mesylate | 22260-51-1 | 99.90% | 1 ML

Supplier: Medchemexpress LLC HY12705A10MM/1ML
Bromocriptine mesylate is a potent dopamine D2/D3 receptor agonist that readily crosses the blood-brain barrier. It stimulates [35S]-GTPγS binding at the D2 dopamine receptor expressed in CHO cells with a pEC50 of 8.15±0.05. It also acts as a strong inhibitor of brain nitric oxide synthase and a potent inhibitor of CYP3A4.
- It is a potent dopamine D2/D3 receptor agonist.
- It is permeable to the blood-brain barrier.
- It shows significant anti-immobility action in experimental models of depression.
- It induces a significant, dose-dependent decrease in pain scores in specific models.
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