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Medchemexpress LLC C26H29F3N4O6S | 2387505-73-7 | 99.7% | 582.59 | 25 MG
Supplier: Medchemexpress LLC 25MGHY111615A
J-2156 TFA is a highly potent, selective somatostatin receptor type 4 (SST4 receptor) agonist. It has IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively. It also demonstrates anti-inflammatory activity and is used for relieving mechanical allodynia and mechanical hyperalgesia in the ipsilateral hindpaws in rats.
- High potency and selectivity for somatostatin receptor type 4 (SST4 receptor)
- IC50 of 0.05 nM for human SST4 and 0.07 nM for rat SST4 receptors
- Possesses anti-inflammatory activity
- Effective in alleviating mechanical allodynia and mechanical hyperalgesia in rats
- Binds with nanomolar affinity to human SST4 (Ki=1.2 nM)
- Over 400-fold subtype-selective against other somatostatin receptors (hsst1, hsst2, hsst3, hsst5)
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