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Medchemexpress LLC C26H29F3N4O6S | 2387505-73-7 | 99.7% | 582.59 | 25 MG
SDP

Catalog No. 5000439187
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J-2156 TFA is a highly potent, selective somatostatin receptor type 4 (SST4 receptor) agonist. It has IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively. It also demonstrates anti-inflammatory activity and is used for relieving mechanical allodynia and mechanical hyperalgesia in the ipsilateral hindpaws in rats.

  • High potency and selectivity for somatostatin receptor type 4 (SST4 receptor)
  • IC50 of 0.05 nM for human SST4 and 0.07 nM for rat SST4 receptors
  • Possesses anti-inflammatory activity
  • Effective in alleviating mechanical allodynia and mechanical hyperalgesia in rats
  • Binds with nanomolar affinity to human SST4 (Ki=1.2 nM)
  • Over 400-fold subtype-selective against other somatostatin receptors (hsst1, hsst2, hsst3, hsst5)

Catalog No. 50-004-39187 Supplier Medchemexpress LLC Supplier No. 25MGHY111615A
May include imposed supplier surcharges.
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J-2156 TFA is a highly potent, selective somatostatin receptor type 4 (SST4 receptor) agonist. It has IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors, respectively. It also demonstrates anti-inflammatory activity and is used for relieving mechanical allodynia and mechanical hyperalgesia in the ipsilateral hindpaws in rats.

  • High potency and selectivity for somatostatin receptor type 4 (SST4 receptor)
  • IC50 of 0.05 nM for human SST4 and 0.07 nM for rat SST4 receptors
  • Possesses anti-inflammatory activity
  • Effective in alleviating mechanical allodynia and mechanical hyperalgesia in rats
  • Binds with nanomolar affinity to human SST4 (Ki=1.2 nM)
  • Over 400-fold subtype-selective against other somatostatin receptors (hsst1, hsst2, hsst3, hsst5)

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