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MilliporeSigma™ Calbiochem™ Adenosine A1 Receptor Agonist II, CCPA

An adenosine analog that acts as a selective, high affinity agonist for Adenosine A1 receptor (A1R) (Ki = 800 pM

Supplier:  MilliporeSigma™ 11913610MG

Catalog No. 11-913-610MG


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Description

Description

An adenosine analog that acts as a selective, high affinity agonist for Adenosine A1 receptor (A1R) (Ki = 800 pM; 2.3μM, 18.8μM, and 42nM for human A1, A2A, A2B, A3 respectively). Shown to be centrally active following systemic administration and exhibits anti-convulsive effects. Also reported to inhibit adenylate cyclase activity in rat fat cell membrane (IC50 = 33nM). Diminishes respiratory rhythm, reduces heart rate, and enhances the activity of KATP channels. Reduces norepinephrine release by about 50% in untreated and pertussis toxin treated hearts.
Specifications

Specifications

White
A1
369.8g/mol
Protect from light
10 mg
99% by HPLC
C15H20ClN5O4
DMSO or H2O
Solid
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