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MilliporeSigma™ Calbiochem™ APT1 Inhibitor II, Cpd21

Catalog No. 5316200001 Shop All MilliporeSigma Products
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53-162-00001 10 mg
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Catalog No. 53-162-00001 Supplier MilliporeSigma™ Supplier No. 5316200001
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Description

A cell permeable acetylpiperazine derivative compound that acts as a selective and reversible inhibitor of lysophospholipase 1 (LYPLA1; IC50 = 840 nM, Ki = 300nM) without affecting the activity of LYPLA2 and 25 other serine hydrolases in mouse BW5147 T cell hydridoma pr

A cell permeable acetylpiperazine derivative compound that acts as a selective and reversible inhibitor of lysophospholipase 1 (LYPLA1; IC50 = 840 nM, Ki = 300nM) without affecting the activity of LYPLA2 and 25 other serine hydrolases in mouse BW5147 T cell hydridoma proteome. Shown to cause an almost complete inhibition (+90%) of LYPLA1 activity in lung, heart, and kidney (50mg/kg, 3 h), and in HEK293T, and mouse T cells (∽ 5μM for 3 h).

Please note that the molecular weight for this compound is batch-specific due to variable water content.
TRUSTED_SUSTAINABILITY

Specifications

Color White
Description 98% by HPLC
Target Proteins APT1
Molecular Formula C18H17ClF3N3O3
Solubility DMSO
Content And Storage Protect from light
Form Solid
Quantity 10 mg
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