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MilliporeSigma™ Calbiochem™ L-745,870 Trihydrochloride

Catalog No. 5058800001 Shop All MilliporeSigma Products
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50-588-00001 10 mg
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Catalog No. 50-588-00001 Supplier MilliporeSigma™ Supplier No. 5058800001
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Description

Selective D4 receptor antagonist with excellent brain penetrat

Selective D4 receptor antagonist with excellent brain penetration. Displays an affinity (Ki) of 0.4nM for human D4 receptors with >1000-fold binding selectivity over D2 and D3 receptors. Does not block agonist-induced activation of GIRK currents. It is used frequently in retinal and CNS studies of D4 modulation.
TRUSTED_SUSTAINABILITY

Specifications

Color Off-white
Description 99% by HPLC
Target Proteins D4
Molecular Formula C18H19N4Cl·3HCl
Solubility H2O
Content And Storage Protect from light
Form Solid
Quantity 10 mg
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