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Medchemexpress LLC Cilastatin-15N,d3 | 2738376-83-3 | 99.7% | C16H23D3N15NO5S | 1 MG
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Supplier:  Medchemexpress LLC HYA0166S1MG

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Cilastatin-15N,d3 is a 15N-labeled and deuterium-labeled form of Cilastatin. Cilastatin (MK0791) acts as a reversible, competitive inhibitor of renal dehydropeptidase I, with an IC50 of 0.1 μM. It also inhibits the bacterial metallo-β-lactamase enzyme CphA at an IC50 of 178 μM. Cilastatin is utilized as an antibacterial adjunct.

  • This compound serves as a tracer.
  • It can be used as an internal standard for quantitative analysis through techniques such as NMR, GC-MS, or LC-MS.
  • The incorporation of stable heavy isotopes (hydrogen, carbon, and other elements) into drug molecules is primarily for quantitation during drug development.
  • Deuteration, in particular, has shown potential to influence the pharmacokinetic and metabolic profiles of drugs.

Catalog No. 50-004-32085


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