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Medchemexpress LLC Cipralisant | 213027-19-1 | 99.3% | 216.32 g/mol | C14H20N2 | 25 MG

Supplier: Medchemexpress LLC HY10699325MG
Cipralisant (GT-2331) is a small-molecule histamine H3 receptor ligand used for research applications. It is reported as a potent, selective, high-affinity H3 receptor full antagonist in vivo and an agonist in vitro, with literature-reported activity values suitable for pharmacological evaluation and click-chemistry applications.
- Potent, high-affinity histamine H3 receptor ligand (pKi ≈ 9.9).
- Shows antagonist activity in vivo and agonist activity in vitro.
- Reported rat H3 Ki ≈ 0.47 nM for target validation studies.
- Contains an alkyne functional group enabling copper-catalyzed azide-alkyne click chemistry.
- High analytical purity (reported ~99.3%), suitable for research use.
- Supplied as a small-scale reagent for pharmacology and AD/HD research.
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