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Medchemexpress LLC CS-VIP 8 hydrochloride | 961.40 | 5 MG

Supplier: Medchemexpress LLC HYP10948A5MG
CS-VIP 8 hydrochloride is a selective allosteric WDR5 protein inhibitor (Kᵢ= 0.008 μM). It induces conformational changes in the MLL1 complex, leading to the dissociation of MLL1 from the complex, inhibiting MLL1 histone methyltransferase activity and regulating HOX gene expression. This compound shows promise for research into hematological diseases like leukemia.
- Selective allosteric WDR5 protein inhibitor (Kᵢ= 0.008 μM).
- Induces conformational changes in the MLL1 complex.
- Leads to the dissociation of MLL1 from the complex.
- Inhibits MLL1 histone methyltransferase activity.
- Regulates HOX gene expression.
- Promising for research into hematological diseases such as leukemia.
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