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Medchemexpress LLC CXCR7 modulator 2 | 2227426-37-9 | 98.7% | 522.68 | 100 MG
SDP

Supplier:  Medchemexpress LLC HY112154100MG

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CXCR7 modulator 2 is a small molecule modulator of C-X-C Chemokine Receptor Type 7 (CXCR7) with a Ki of 13 nM. This compound exhibits potent CXCR7-binding affinity and β-arrestin activity, offering improved selectivity in GPCR panels and an enhanced therapeutic index in hERG patch-clamp assays. It demonstrates good aqueous solubility and is suitable for research applications.

  • Potent CXCR7-binding affinity (Ki=13 nM)
  • Beta-arrestin activity (EC50=11 nM)
  • Improved selectivity in GPCR panel
  • Improved therapeutic index in hERG patch-clamp assay
  • Moderate to high in vitro turnover
  • Good aqueous solubility
  • Rapidly absorbed in vivo
  • Reduces cardiac fibrosis in injury models
  • Soluble in DMSO

Catalog No. 50-004-37958


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