Learn More
Medchemexpress LLC Dagrocorat | 1044535-52-5 | 99.9% | 494.55 | 50 MG

Supplier: Medchemexpress LLC HY1671850MG
Dagrocorat (PF-00251802) is an orally active and selective high-affinity partial agonist of the glucocorticoid receptor. It is also a time-dependent reversible inhibitor of CYP3A (IC50=1.3 μM in human liver microsomes) and CYP2D6 (Ki=0.57 μM in human liver microsomes). It can be used for the research of rheumatoid arthritis.
- Orally active and selective high-affinity partial agonist of the glucocorticoid receptor.
- Time-dependent reversible inhibitor of CYP3A (IC50=1.3 μM in human liver microsomes) and CYP2D6 (Ki=0.57 μM in human liver microsomes).
- Can be used for the research of rheumatoid arthritis.
By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.