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Medchemexpress LLC Dagrocorat (PF-00251802) | 1044535-52-5 | 99.9% | 494.55 g/mol | C29H29F3N2O2 | 10 MG

Supplier: Medchemexpress LLC HY1671810MG
Dagrocorat (PF-00251802) is an orally active, selective, high-affinity partial agonist of the glucocorticoid receptor supplied for research use. It exhibits time-dependent reversible inhibition of CYP3A and inhibitory activity against CYP2D6, and is used in preclinical studies of inflammatory conditions such as rheumatoid arthritis.
- Orally active glucocorticoid receptor partial agonist useful for mechanistic studies.
- Shows time-dependent reversible inhibition of CYP3A and inhibits CYP2D6 (IC50/Ki values reported).
- High chemical purity (99.9%) suitable for research applications.
- Provided in small research quantities (10 MG) for laboratory use.
- Solid form with reported solubility in common organic solvents; follow supplier documentation for handling.
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