Cayman Chemical DIlazephydrochlorIde 10mg

Supplier:  Cayman Chemical 2976110 MG

An ENT1 inhibitor (IC50 = 17.5 nM); selective for ENT1 over ENT2 (IC50 = 8,800 nM); increases adenosine-induced relaxation of isolated guinea pig taenia caeci strips at 0.03 and 0.3 µM; decreases calcium-induced contractions in isolated guinea pig taenia caeci strips at 1, 5, and 10 µM; reduces heart rate and systolic, mean, and diastolic aortic pressure and increases left ventricular blood flow in anesthetized dogs at 0.2 mg/kg, i.v.; reduces aortic platelet adhesion and aggregation in a rabbit model of aortic injury-induced thrombosis at 0.1 mg/kg

Catalog No. 50-298-9184