Medchemexpress LLC Dopamine D2 receptor agonist-3 | 1257326-24-1 | 98.3% | 295.81 g/mol | C15H22ClN3O | 25 MG

Supplier:  Medchemexpress LLC HY10341825MG

Dopamine D2 receptor agonist-3 is a research compound characterized as a selective D2 receptor partial agonist and a D3 receptor antagonist. In vitro activity is reported with pEC50 8.3 at D2 and <5.5 at D3. In vivo, a 3 mg/kg (s.c.) dose demonstrated high brain penetration (brain:blood ratio ≈5.5) with Tmax ≈0.5 h. The compound is a solid with reported purity of 98.3% and molecular formula C15H22ClN3O.

• Selective D2 receptor partial agonist and D3 receptor antagonist.
• Reported pEC50 values: 8.3 (D2) and <5.5 (D3).
• High reported purity (98.3%).
• Solid form, suitable for research applications.
• Demonstrated brain penetration in vivo (3 mg/kg, s.c.; brain:blood ratio ~5.5).
• Available in small pack sizes, including 25 mg.

Catalog No. 50-002-45145