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Medchemexpress LLC DS-1971a | 1450595-86-4 | 99.3% | 50 MG

Supplier: Medchemexpress LLC HY13118250MG
DS-1971a is a potent, selective, and orally active NaV1.7 inhibitor, with IC50s of 22.8 nM for hNaV1.7 and 59.4 nM for mNaV1.7. It exerts analgesic effects and addresses thermal hyperalgesia and mechanical hypersensitivity.
- Potent, selective, and orally active NaV1.7 inhibitor
- Inhibitory concentration (IC50) of 22.8 nM for hNaV1.7
- Exerts analgesic effects
- Soluble in DMSO at 100 mg/mL
- Powder stable for 3 years at -20°C and 2 years at 4°C
- Stable in solvent for 2 years at -80°C and 1 year at -20°C
- Targets sodium channel membrane transporter/ion channel
- Exhibits a favorable toxicological profile
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