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Medchemexpress LLC (E/Z)-4-Hydroxytamoxifen (Afimoxifene) | 68392-35-8 | 99.6% | 387.51 | 5 MG

Supplier: Medchemexpress LLC HY16950A5MG
(E/Z)-4-Hydroxytamoxifen (Afimoxifene) is a racemic compound consisting of (Z)-4-Hydroxytamoxifen and (E)-4-Hydroxytamoxifen isomers. It acts as a selective estrogen receptor modulator with both estrogenic and antiestrogenic activities and is an active metabolite of Tamoxifen.
- Acts as a selective estrogen receptor modulator with both estrogenic and antiestrogenic activities.
- Is an active metabolite of Tamoxifen.
- Acts as an agonist of the G protein-coupled estrogen receptor (GPER) with relatively low affinity (100-1000 nM).
- Shows promise for research into cyclical mastalgia, including breast pain, tenderness, and nodularity.
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