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Medchemexpress LLC Efaroxan hydrochloride | 89197-00-2 | 99.80% | 25 MG

Supplier: Medchemexpress LLC 25MGHYB1416A
Efaroxan hydrochloride is a potent, selective, and orally active α2-adrenoceptor antagonist, demonstrating antidiabetic activity. It also acts as a selective I1-Imidazoline receptor antagonist. This compound can be utilized in research related to cardiovascular disease.
- Potent, selective, and orally active α2-adrenoceptor antagonist.
- Possesses antidiabetic activity.
- Selective I1-Imidazoline receptor antagonist.
- Applicable for research in cardiovascular disease.
- Binds to I1-imidazoline and α2-adrenergic receptors with Kᵢ values of 0.15 nM and 5.6 nM, respectively, in bovine rostral ventrolateral medulla membranes.
- Increases plasma insulin levels in conscious fed and fasted rats without significantly affecting plasma glucose levels.
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