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Medchemexpress LLC Endomorphin 1 acetate | 1276123-71-7 | 99.9% | 670.75 | 25 MG
Supplier: Medchemexpress LLC 25MGHYP0185A
Endomorphin 1 acetate is a highly selective agonist of the μ-opioid receptor (Ki: 1.11 nM). It also shows reasonable affinities for kappa3 binding sites with a Ki value between 20 and 30 nM. This compound possesses antinociceptive properties.
- Highly selective agonist of the μ-opioid receptor (Ki: 1.11 nM)
- Displays reasonable affinities for kappa3 binding sites (Ki between 20 and 30 nM)
- Inhibits Forskolin-stimulated cyclic AMP formation
- Increases interleukin-8 secretion in Caco-2 cells
- Inhibits excitatory transmission in adult rat substantia gelatinosa neurons
- Exhibits antinociceptive properties in mice
- Alleviates myocardial ischemia/reperfusion injury in rats
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