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Medchemexpress LLC Ensitrelvir fumarate | 2757470-18-9 | 100.0% | C26H21ClF3N9O6 | 50 MG
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Supplier:  Medchemexpress LLC HY143216A50MG

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Ensitrelvir fumarate, also known as S-217622 fumarate, is the first orally active, non-covalent, and non-peptidic SARS-CoV-2 3CL protease inhibitor with an IC50 of 13 nM. It demonstrates significant antiviral activity against various SARS-CoV-2 variants, SARS-CoV, and MERS-CoV.

  • First orally active, non-covalent, non-peptidic SARS-CoV-2 3CL protease inhibitor
  • Inhibits SARS-CoV-2 3CL protease with an IC50 of 13 nM
  • Effective against wild-type SARS-CoV-2 and Alpha, Beta, Gamma, and Delta variants with EC50 values around 0.4 μM
  • Shows EC50 values of 0.21 μM for SARS-CoV and 1.4 μM for MERS-CoV
  • Dose-dependently inhibits intrapulmonary replication of SARS-CoV-2 in mice

Catalog No. 50-003-53833


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