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Medchemexpress LLC Ensitrelvir fumarate | 2757470-18-9 | 99.99% | C26H21ClF3N9O6 | 1 ML
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Supplier:  Medchemexpress LLC HY143216A10MM/1ML

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Ensitrelvir (S-217622) fumarate is the first orally active, non-covalent, non-peptidic SARS-CoV-2 3CL protease inhibitor. It demonstrates high potency with an IC50 of 13 nM and is intended for research use only. The compound has shown significant antiviral activity in vitro against various SARS-CoV-2 variants.

  • First orally active, non-covalent, non-peptidic SARS-CoV-2 3CL protease inhibitor.
  • Exhibits an IC50 of 13 nM, indicating high potency.
  • Effective against wild-type SARS-CoV-2 and Alpha, Beta, Gamma, and Delta variants with EC50 values of approximately 0.4 μM.
  • Also active against SARS-CoV and MERS-CoV, with EC50 values of 0.21 and 1.4 μM, respectively.
  • Dose-dependently inhibits intrapulmonary replication of SARS-CoV-2 in mice.

Catalog No. 50-003-54749


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