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Medchemexpress LLC Estra-1,3,5(10)-triene-3,17-diol (17β)-, 3-sulfamate | 172377-52-5 | MFCD00947822 | 351.46 | 100 MG
Supplier: Medchemexpress LLC HYU00112100MG
Estradiol 3-sulfamate, also known as E2MATE, is a potent, long-acting, and orally active steroid sulfatase inhibitor. It effectively inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. This compound is transformed and absorbed in the gut into its oxidative metabolite, EMATE, both of which are strong steroid sulfatase inhibitors. It is intended for research use only.
- Potent, long-acting steroid sulfatase inhibitor
- Orally active
- Inhibits estrone sulfatase (IC50 of 251 nM)
- Shows growth inhibitory effects on various cancer cell lines
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