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Medchemexpress LLC Estradiol 3-sulfamate | 172377-52-5 | 351.46 | 50 MG
SDP

Catalog No. 5000448429
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Estradiol 3-sulfamate is a potent, long-acting, and orally active steroid sulfatase inhibitor. It inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. The compound is readily transformed and absorbed in the gut into its oxidative metabolite, EMATE, demonstrating potent and long-acting STS inhibition.

  • Potent, long-acting, and orally active steroid sulfatase inhibitor.
  • Inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM.
  • Increased estrone sulfatase inhibitory activity with specific halogen moieties.
  • Readily absorbed and transformed in the gut into its oxidative metabolite, EMATE.
  • Both compounds demonstrate potent and long-acting STS inhibition.

Catalog No. 50-004-48429 Supplier Medchemexpress LLC Supplier No. HYU0011250MG
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Estradiol 3-sulfamate is a potent, long-acting, and orally active steroid sulfatase inhibitor. It inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. The compound is readily transformed and absorbed in the gut into its oxidative metabolite, EMATE, demonstrating potent and long-acting STS inhibition.

  • Potent, long-acting, and orally active steroid sulfatase inhibitor.
  • Inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM.
  • Increased estrone sulfatase inhibitory activity with specific halogen moieties.
  • Readily absorbed and transformed in the gut into its oxidative metabolite, EMATE.
  • Both compounds demonstrate potent and long-acting STS inhibition.

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