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Medchemexpress LLC EZM0414 | 2411748-50-8 | 99.1% | C22H29FN4O2 | 50 MG
Supplier: Medchemexpress LLC HY14485850MG
EZM0414 is a potent, selective, and orally bioavailable inhibitor of SETD2. It is used for the research of relapsed or refractory multiple myeloma and diffuse large B-cell lymphoma.
- Potent, selective, orally bioavailable inhibitor of SETD2
- IC50 of 18 nM in SETD2 biochemical assay
- IC50 of 34 nM in cellular assay
- Inhibits proliferation of MM and DLBCL cell lines
- Well-tolerated and inhibits tumor growth in xenograft models
- Almost 100% oral bioavailability in rats and mice
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